PI3Kα-IN-22 is a potent WT-sparing, PI3Kα(H1047R) inhibitor, designed to target specific mutations, which serves as a driver oncogene in certain cancers. This particular compound was recently highlighted by the Drug Hunter. 


We have selected a set of PI3Kα inhibitor analogs that are readily available to enrich your research. 


Also, we at Chemspace provide comprehensive Discovery Solutions! We will navigate you through accessible chemical space using our computational approaches to identify new chemotypes for the target of interest.   

Chemspace – your end-to-end Discovery CRO.