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IUPAC Name:

(1S,2S,10R,18R)-6-(4-chlorophenyl)-19-(cyclopropylmethyl)-2-methoxy-11-oxa-8,19-diazahexacyclo[10.9.1.0¹,¹⁰.0²,¹⁸.0⁴,⁹.0¹⁶,²²]docosa-4(9),5,7,12,14,16(22)-hexaen-13-ol

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MedChemExpress Ships from: United States To:	TBD	POA	1 mg	Go to cart Enquire
Description: Names: SRI-22136; Product Description: SRI-22136 is a Delta Opioid Receptor (DOR) antagonist that can cross blood-brain barrier with a IC50 of 0.42 nM. SRI-22136 does not have agonistic activity but antagonistic activity against DOR, MOR (IC50 = 370 nM), KOR (IC50 = 54 nM) and can avoid addiction/aversion effects. SRI-22136 can effectively inhibit the BACE1 activity induced by DADLE (a DOR agonist) (HY-105343) (IC50 = 120 nM). SRI-22136 prevents completely Alzheimer’s-like pathology in mouse model. SRI-22136 can used for the study of Alzheimer’s disease; Target: Beta-secretase;Opioid Receptor
MedChemExpress EU Ships from: Sweden To:	TBD	POA	1 mg	Go to cart Enquire
Description: Names: SRI-22136; Product Description: SRI-22136 is a Delta Opioid Receptor (DOR) antagonist that can cross blood-brain barrier with a IC50 of 0.42 nM. SRI-22136 does not have agonistic activity but antagonistic activity against DOR, MOR (IC50 = 370 nM), KOR (IC50 = 54 nM) and can avoid addiction/aversion effects. SRI-22136 can effectively inhibit the BACE1 activity induced by DADLE (a DOR agonist) (HY-105343) (IC50 = 120 nM). SRI-22136 prevents completely Alzheimer’s-like pathology in mouse model. SRI-22136 can used for the study of Alzheimer’s disease; Target: Beta-secretase;Opioid Receptor

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Zoom the structure CSCS21121923909 Add to cart

IUPAC Name:

N-[(1S,5R,13R,14S,17S)-4-(cyclopropylmethyl)-10,17-dihydroxy-12-oxa-4-azapentacyclo[9.6.1.0¹,¹³.0⁵,¹⁷.0⁷,¹⁸]octadeca-7(18),8,10-trien-14-yl]-1H-pyrrolo[2,3-c]pyridine-7-carboxamide hydrochloride

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MedChemExpress Ships from: United States To:	TBD	POA	1 mg	Go to cart Enquire
Description: Names: MOR antagonist 2 (hydrochloride); Product Description: MOR antagonist 2 hydrochloride is a blood-brain barrier-permeable μ-opioid receptor (MOR) antagonist, with an IC50 of 28.37 nM, an EC50 of 4.25 nM, and a Ki of 0.18 nM against MOR. MOR antagonist 2 hydrochloride stabilizes the inactive conformation of MOR to reduce receptor activation levels. MOR antagonist 2 hydrochloride antagonizes analgesic effects in the mouse warm-water tail-flick test. MOR antagonist 2 hydrochloride induces fewer opioid withdrawal symptoms (wet dog shakes, paw tremors) in mice with opioid withdrawal symptoms. MOR antagonist 2 hydrochloride can be used for the research of opioid use disorder; Target: Opioid Receptor; CAS: 3075862-29-9
MedChemExpress EU Ships from: Sweden To:	TBD	POA	1 mg	Go to cart Enquire
Description: Names: MOR antagonist 2 (hydrochloride); Product Description: MOR antagonist 2 hydrochloride is a blood-brain barrier-permeable μ-opioid receptor (MOR) antagonist, with an IC50 of 28.37 nM, an EC50 of 4.25 nM, and a Ki of 0.18 nM against MOR. MOR antagonist 2 hydrochloride stabilizes the inactive conformation of MOR to reduce receptor activation levels. MOR antagonist 2 hydrochloride antagonizes analgesic effects in the mouse warm-water tail-flick test. MOR antagonist 2 hydrochloride induces fewer opioid withdrawal symptoms (wet dog shakes, paw tremors) in mice with opioid withdrawal symptoms. MOR antagonist 2 hydrochloride can be used for the research of opioid use disorder; Target: Opioid Receptor; CAS: 3075862-29-9
Targetmol Chemicals Inc Ships from: United States To:	TBD	POA	1 mg	Go to cart Enquire
Description: MOR antagonist 2 hydrochloride is a μ-opioid receptor (MOR) antagonist that can cross the blood-brain barrier. It exhibits an IC₅₀ of 28.37 nM, an EC50 of 4.25 nM, and a Ki of 0.18 nM at MOR. This compound stabilizes the inactive conformation of MOR, thereby reducing receptor activation levels. In mice, MOR antagonist 2 hydrochloride counteracts analgesic effects in the warm-water tail-flick test and induces fewer opioid withdrawal symptoms, such as wet-dog shakes and paw tremors. It is applicable in researching opioid use disorder.; CAS: 3075862-29-9

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Zoom the structure CSCS21383945598 Add to cart

IUPAC Name:

N-{2-[1-(6-bromonaphthalene-2-carbonyl)-3-hydroxypiperidin-3-yl]ethyl}-6-chloro-4-fluoro-1H-indole-2-carboxamide

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Enamine Ltd. Ships from: Ukraine To:	TBD	POA	1 mg	Go to cart Enquire

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Zoom the structure CSCS14831850878 Add to cart

IUPAC Name:

(1S,2S,13R,21R)-11-benzyl-22-(cyclopropylmethyl)-14-oxa-11,22-diazaheptacyclo[13.9.1.0¹,¹³.0²,²¹.0⁴,¹².0⁵,¹⁰.0¹⁹,²⁵]pentacosa-4(12),5,7,9,15(25),16,18-heptaene-2,16-diol hydrochloride

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Targetmol Chemicals Inc Ships from: United States To:	30 days	1,820.00		Go to cart Enquire
Description: δ2 opioid receptor antagonist; CAS: 1206487-81-1
Key Organics Limited (BIONET) Ships from: United Kingdom To:	TBD	POA	1 mg	Go to cart Enquire
MedChemExpress Ships from: United States To:	TBD	POA	1 mg	Go to cart Enquire
Description: Names: N-Benzylnaltrindole (hydrochloride); Product Description: N-Benzylnaltrindole hydrochloride is a potent δ2-selective opioid receptor antagonist. Benzylnaltrindole hydrochloride has a long duration of action in vivo than Naltriben (NTB). N-Benzylnaltrindole hydrochloride iserve as a useful tool in the pharmacologic characterization of δ-opioid receptor function; Target: Opioid Receptor; CAS: 1206487-81-1
MedChemExpress EU Ships from: Sweden To:	TBD	POA	1 mg	Go to cart Enquire
Description: Names: N-Benzylnaltrindole (hydrochloride); Product Description: N-Benzylnaltrindole hydrochloride is a potent δ2-selective opioid receptor antagonist. Benzylnaltrindole hydrochloride has a long duration of action in vivo than Naltriben (NTB). N-Benzylnaltrindole hydrochloride iserve as a useful tool in the pharmacologic characterization of δ-opioid receptor function; Target: Opioid Receptor; CAS: 1206487-81-1

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Zoom the structure CSCS00102514306 Add to cart

IUPAC Name:

(1R,2S,13R,21R)-11-benzyl-22-(cyclopropylmethyl)-14-oxa-11,22-diazaheptacyclo[13.9.1.0¹,¹³.0²,²¹.0⁴,¹².0⁵,¹⁰.0¹⁹,²⁵]pentacosa-4(12),5,7,9,15(25),16,18-heptaene-2,16-diol hydrochloride

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Apexbio Technology LLC Ships from: United States To:	40 days	216.70		Go to cart Enquire
Description: Name: N-Benzylnaltrindole hydrochloride; δ2 opioid receptor antagonist; Format: white crystalline solid; CAS: 1206487-81-1

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Zoom the structure CSCS03436517393 Add to cart

IUPAC Name:

(1S,2S,13R)-11-benzyl-22-(cyclopropylmethyl)-14-oxa-11,22-diazaheptacyclo[13.9.1.0¹,¹³.0²,²¹.0⁴,¹².0⁵,¹⁰.0¹⁹,²⁵]pentacosa-4(12),5,7,9,15(25),16,18-heptaene-2,16-diol hydrochloride

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Angene International Limited Ships from: China To:	TBD	POA	1 g	Go to cart Enquire
Description: N-BENZYLNALTRINDOLE HYDROCHLORIDE; CAS: 1206487-81-1
Angene US Ships from: United States To:	TBD	POA	1 g	Go to cart Enquire
Description: N-BENZYLNALTRINDOLE HYDROCHLORIDE; CAS: 1206487-81-1

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Zoom the structure CSCS14813048497 Add to cart

IUPAC Name:

(1S,2S,3S,4S,5R,6S,8S,9S,10R,13S,16S,17S)-11-ethyl-3,8-dihydroxy-4,6,16-trimethoxy-11-azahexacyclo[7.7.2.1²,⁵.0¹,¹⁰.0³,⁸.0¹³,¹⁷]nonadecan-13-yl 2-acetamidobenzoate hydrochloride

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10X CHEM Ships from: United States To:	TBD	POA	1 g	Go to cart Enquire
Description: Lappaconitine HCl; CAS: 767350-42-5
Targetmol Chemicals Inc Ships from: United States To:	TBD	POA	1 mg	Go to cart Enquire
Description: Lappaconitine HCl is a centrally acting non-opioid analgesic and class-I antiarrhythmic. It acts by binding to the site-2 receptor and irreversibly blocking hH1 sodium channels.; CAS: 767350-42-5

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Zoom the structure CSCS06595022588 Add to cart

IUPAC Name:

(1S,5R,13R,14S,17S)-14-(2,5,8,11,14,17-hexaoxanonadecan-19-yloxy)-10-methoxy-4-methyl-12-oxa-4-azapentacyclo[9.6.1.0¹,¹³.0⁵,¹⁷.0⁷,¹⁸]octadeca-7,9,11(18)-trien-17-ol hydrochloride

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Targetmol Chemicals Inc Ships from: United States To:	30 days	1,970.00		Go to cart Enquire
Description: Oxicodegol HCl is a mu-opioid agonist used in the treatment of Moderate to Severe Chronic Low Back Pain; CAS: 1211231-53-6

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Zoom the structure CSCS14948337563 Add to cart

IUPAC Name:

4-{[(2R,7aS)-2-fluoro-hexahydro-1H-pyrrolizin-7a-yl]methoxy}-15-chloro-28-fluoro-1,3,5,9-tetraazapentacyclo[21.3.1.1⁶,¹⁰.0²,⁷.0¹¹,¹⁶]octacosa-2,4,6(28),7,9,11,13,15-octaene-13,23-diol

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Targetmol Chemicals Inc Ships from: United States To:	30 days	2,720.00		Go to cart Enquire
Description: KRAS inhibitor-25 (compound 151a), a pyrido[2,3-d]pyrimidine derivative, effectively inhibits KRas G12V, KRas WT, and KRas G12R with IC₅₀ values all below 100 nM.; CAS: 3030577-05-7
MedChemExpress Ships from: United States To:	TBD	POA	1 mg	Go to cart Enquire
Description: Names: KRAS inhibitor-25; Product Description: KRAS inhibitor-25 (compound 151a) is a pyridopyrimidine KRAS inhibitor, with an IC50 of ; Target: Ras; CAS: 3030577-05-7
MedChemExpress EU Ships from: Sweden To:	TBD	POA	1 mg	Go to cart Enquire
Description: Names: KRAS inhibitor-25; Product Description: KRAS inhibitor-25 (compound 151a) is a pyridopyrimidine KRAS inhibitor, with an IC50 of ; Target: Ras; CAS: 3030577-05-7

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Zoom the structure CSCS20591796832 Add to cart

IUPAC Name:

(14Z)-14-{2-[(14Z)-10,17-dihydroxy-4-(prop-2-en-1-yl)-12-oxa-4-azapentacyclo[9.6.1.0¹,¹³.0⁵,¹⁷.0⁷,¹⁸]octadeca-7,9,11(18)-trien-14-ylidene]hydrazin-1-ylidene}-4-(prop-2-en-1-yl)-12-oxa-4-azapentacyclo[9.6.1.0¹,¹³.0⁵,¹⁷.0⁷,¹⁸]octadeca-7,9,11(18)-triene-10,17-diol dihydrochloride

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Targetmol Chemicals Inc Ships from: United States To:	30 days	178.00		Go to cart Enquire
Description: μ1 receptor antagonist; CAS: 880759-65-9

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Zoom the structure CSCS03437860595 Add to cart

IUPAC Name:

14-{2-[10,17-dihydroxy-4-(prop-2-en-1-yl)-12-oxa-4-azapentacyclo[9.6.1.0¹,¹³.0⁵,¹⁷.0⁷,¹⁸]octadeca-7,9,11(18)-trien-14-ylidene]hydrazin-1-ylidene}-4-(prop-2-en-1-yl)-12-oxa-4-azapentacyclo[9.6.1.0¹,¹³.0⁵,¹⁷.0⁷,¹⁸]octadeca-7,9,11(18)-triene-10,17-diol dihydrochloride

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Biosynth Ships from: United Kingdom To:	30 days	990.00	25 mg	Go to cart Enquire
Description: Naloxonazine dihydrochloride; CAS: 880759-65-9

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Zoom the structure CSCS02125604652 Add to cart

IUPAC Name:

(1S,5R,13S,14Z,17S)-14-{2-[(1S,5R,13S,14E,17S)-10,17-dihydroxy-4-(prop-2-en-1-yl)-12-oxa-4-azapentacyclo[9.6.1.0¹,¹³.0⁵,¹⁷.0⁷,¹⁸]octadeca-7,9,11(18)-trien-14-ylidene]hydrazin-1-ylidene}-4-(prop-2-en-1-yl)-12-oxa-4-azapentacyclo[9.6.1.0¹,¹³.0⁵,¹⁷.0⁷,¹⁸]octadeca-7,9,11(18)-triene-10,17-diol dihydrochloride

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Apexbio Technology LLC Ships from: United States To:	40 days	190.30		Go to cart Enquire
Description: Name: Naloxonazine dihydrochloride; μ1 receptor antagonist; Format: off-white solid; CAS: 880759-65-9

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Zoom the structure CSCS03436517395 Add to cart

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